With the help of Light Microscope, Scanning Electron Microscope (SEM) and Transmission Electron Microscope (TEM), comparative observation was made into the impact of Binds Dissipating Tablet on ultra-microstructure of transplanted Hepatoma Carcinoma Cell (HCC) of mice and the anticancer mechanism. Results have shown the tablet directly killed or seriously damaged HCC through direct action on HCC membrane and produced immediate and long-acting breakdown of HCC with short-term application.