Traditional Chinese medicine (TCM) is the basic element of the formula, and the embodiment of the implementation of treatment is based on syndrome differentiation in TCM. The understanding of Chinese medicinals determines the clinical curative effect. It is of great practical significance to collect and excavate China′s ancient classics about traditional Chinese medicine. At present, there is more in-depth understanding and research on ancient books of traditional Chinese medicine, classics of traditional Chinese medicine of ethnic minorities and the Buddhist classics medicine, but less research on the traditional Chinese medicine in the Taoist classic series, Taoist canon. Based on Taiping Part of Taoist canon in Ming dynasty, this study collected and explored the Chinese medicinals part so as to provide references for modern medicine research and application.